Kinetics of human cannabinoid 1 (CB1) receptor antagonists: Structure-kinetics relationships (SKR) and implications for insurmountable antagonism
Lizi Xia, Henk de Vries, Xue Yang, Eelke B Lenselink, Athina Kyrizaki, Francis Barth, Julien Louvel, Matthias K Dreyer, Daan van der Es, Adriaan P IJzerman, Laura H Heitman
Biochemical Pharmacology, 151, 166-179 (2018) .
2018
Full text: http://dx.doi.org/10.1016/j.bcp.2017.10.014
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