Rational design of a novel peripherally-restricted, orally active CB1 cannabinoid antagonist containing a 2,3-diarylpyrrole motif
Laurent Hortala, Murielle Rinaldi-Carmona, Christian Congy, Laurent Boulu, Freddy Sadoun, Gérard Fabre, Olivier Finance, Francis Barth
Bioorganic & Medicinal Chemistry Letters, 20(15), 4573–4577 (2010) .
2010
Full text: http://dx.doi.org/10.1016/j.bmcl.2010.06.017
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